Listar Artículos (Farmacología) por autor "Burgos Morón, Estefanía"
Mostrando ítems 1-20 de 22
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5-Aza-2'-deoxycytidine causes replication lesions that require Fanconi anemia-dependent homologous recombination for repair
Orta Vázquez, Manuel Luis; Calderón Montaño, José Manuel; Domínguez García, Inmaculada; Pastor Carrillo, Nuria María; Burgos Morón, Estefanía; López Lázaro, Miguel; Cortés, Felipe; Mateos Cordero, Santiago; Helleday, Thomas (Oxford University Press, 2013)5-Aza-2'-deoxycytidine (5-azadC) is a DNA methyltransferase (DNMT) inhibitor increasingly used in treatments of hematological ...
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A hydroalcoholic extract from the leaves of Nerium oleander inhibits glycolysis and induces selective killing of lung cancer cells
Calderón Montaño, José Manuel; Burgos Morón, Estefanía; Orta Vázquez, Manuel Luis; Mateos Cordero, Santiago; López Lázaro, Miguel (Georg Thieme Verlag, 2013)Recent evidence suggests that cardiac glycosides might be used for the treatment of cancer. The ornamental shrub Nerium ...
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Artificial Diets Based on Selective Amino Acid Restriction versus Capecitabine in Mice with Metastatic Colon Cancer
Jiménez Alonso, Julio José; Guillén Mancina, Emilio; Calderón Montaño, José Manuel; Jiménez González, Víctor; Díaz Ortega, Patricia; Burgos Morón, Estefanía; López Lázaro, Miguel (MDPI, 2022)New therapies are needed to improve the low survival rates of patients with metastatic colon cancer. Evidence suggests ...
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Artificial Diets with Altered Levels of Sulfur Amino Acids Induce Anticancer Activity in Mice with Metastatic Colon Cancer, Ovarian Cancer and Renal Cell Carcinoma
Jiménez Alonso, Julio José; Guillén Mancina, Emilio; Calderón Montaño, José Manuel; Jiménez González, Víctor; Díaz Ortega, Patricia; Burgos Morón, Estefanía; López Lázaro, Miguel (Multidisciplinary Digital Publishing Institute (MDPI), 2023)Sulfur-containing amino acids methionine (Met), cysteine (Cys) and taurine (Tau) are common dietary constituents with ...
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Artificial Diets with Selective Restriction of Amino Acids and Very Low Levels of Lipids Induce Anticancer Activity in Mice with Metastatic Triple-Negative Breast Cancer
Guillén Mancina, Emilio; Jiménez Alonso, Julio José; Calderón Montaño, José Manuel; Jiménez González, Víctor; Díaz Ortega, Patricia; Burgos Morón, Estefanía; López Lázaro, Miguel (Multidisciplinary Digital Publishing Institute (MDPI), 2023)Current treatments for patients with metastatic triple negative breast cancer (TNBC) are generally ineffective. This ...
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Cells Deficient in the Fanconi Anemia Protein FANCD2 are Hypersensitive to the Cytotoxicity and DNA Damage Induced by Coffee and Caffeic Acid
Burgos Morón, Estefanía; Calderón Montaño, José Manuel; Orta Vázquez, Manuel Luis; Guillén Mancina, Emilio; Mateos Cordero, Santiago; López Lázaro, Miguel (MDPI AG, 2016)Epidemiological studies have found a positive association between coffee consumption and a lower risk of cardiovascular ...
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Comment on ‘Quiescence and γH2AX in neuroblastoma are regulated by Ouabain/Na,K-ATPase': ouabain and cáncer
Calderón Montaño, José Manuel; Burgos Morón, Estefanía; López Lázaro, Miguel (Nature Publishing Group, 2013) -
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Consumption of the Dietary Flavonoids Quercetin, Luteolin and Kaempferol and Overall Risk of Cancer - A Review and Meta-Analysis of the Epidemiological Data
López Lázaro, Miguel; Burgos Morón, Estefanía; Tena, J.D.; Sanz, I.; Sainz, J; Calderón Montaño, José Manuel (Biomedical Publisher, 2013)Numerous epidemiological and preclinical studies suggest that flavonoids may play an important role in the decreased risk ...
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Dichloroacetate, 2-Deoxyglucose and a Hydroalcoholic Extract from the Skin of the Fruit of Solanum melongena (Aubergine) Induce Selective Anticancer Activity against Melanoma Cells
Calderón Montaño, José Manuel; Burgos Morón, Estefanía; Martínez Sánchez, Sara María; López Lázaro, Miguel (Biomedical Publisher, 2013)Prognosis of melanoma patients with metastatic disease is very poor. For example, over 95% of melanoma patients with three ...
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Effect of DNA repair deficiencies on the cytotoxicity of resveratrol
López Lázaro, Miguel; Burgos Morón, Estefanía; Calderón Montaño, José Manuel; Orta Vázquez, Manuel Luis; Mateos Cordero, Santiago (2015)Numerous preclinical studies have shown that the naturally-occurring polyphenol resveratrol may produce health-beneficial ...
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Evaluating the cancer therapeutic potential of cardiac glycosides
Calderón Montaño, José Manuel; Burgos Morón, Estefanía; Orta Vázquez, Manuel Luis; Maldonado Navas, Dolores; García Domínguez, Irene; López Lázaro, Miguel (Hindawi Publishing Corporation, 2014)Cardiac glycosides, also known as cardiotonic steroids, are a group of natural products that share a steroid-like structure ...
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In vitro anticancer activity and mechanism of action of an aziridinyl galactopyranoside
Burgos Morón, Estefanía; Pastor Carrillo, Nuria María; Orta Vázquez, Manuel Luis; Jiménez Alonso, Julio José; Palo Nieto, Juan Carlos; Vega Holm, Margarita; Vega Pérez, José Manuel; Iglesias Guerra, Fernando; Mateos Cordero, Santiago; López Lázaro, Miguel; Calderón Montaño, José Manuel (Multidisciplinary Digital Publishing Institute (MDPI), 2022)We recently screened a series of new aziridines β-D-galactopyranoside derivatives for selective anticancer activity and ...
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Manipulation of Amino Acid Levels with Artificial Diets Induces a Marked Anticancer Activity in Mice with Renal Cell Carcinoma
Calderón Montaño, José Manuel; Guillén Mancina, Emilio; Jiménez Alonso, Julio José; Jiménez González, Víctor; Burgos Morón, Estefanía; Mate Barrero, Alfonso; Pérez Guerrero, María Concepción; López Lázaro, Miguel (Multidisciplinary Digital Publishing Institute (MDPI), 2022)Targeted therapies with antiangiogenic drugs (e.g., sunitinib) and immune checkpoint inhibitors (e.g., anti-PD-1 antibodies) ...
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Repurposing Study of 4-Acyl-1-phenylaminocarbonyl-2-substituted-piperazine Derivatives as Potential Anticancer Agents-In Vitro Evaluation against Breast Cancer Cells
Guillén Mancina, Emilio; García Lozano, María del Rosario; Burgos Morón, Estefanía; Mazzotta, Sarah; Martínez Aguado, Pablo; Calderón Montaño, José Manuel; Vega Pérez, José Manuel; López Lázaro, Miguel; Iglesias Guerra, Fernando; Vega Holm, Margarita (MDPI, 2023)first_pagesettingsOrder Article Reprints Open AccessArticle Repurposing Study of 4-Acyl-1-phenylaminocarbonyl-2-substituted-piperazine ...
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Role of the Intracellular pH in the Metabolic Switch between Oxidative Phosphorylation and AerobicGlycolysis - Relevance to Cancer
Calderón Montaño, José Manuel; Burgos Morón, Estefanía; Pérez Guerrero, María Concepción; Salvador Bofill, Francisco Javier; Robles Frías, Antonio; López Lázaro, Miguel (Biomedical Publisher, 2011)Cellular energy in the form of ATP can be produced through oxidative phosphorylation and through glycolysis. Since ...
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Screening for selective anticancer activity of 65 extracts of plants collected in Western Andalusia, Spain
Calderón Montaño, José Manuel; Martínez Sánchez, Sara María; Jiménez González, Víctor; Burgos Morón, Estefanía; Guillén Mancina, Emilio; Jiménez Alonso, Julio José; Díaz Ortega, Patricia; García Martín, Felipe José; Aparicio Martínez, Abelardo; López Lázaro, Miguel (Multidisciplinary Digital Publishing Institute (MDPI), 2021)Finding cytotoxic drugs with a high selectivity towards cancer cells is crucial to improve the low survival rates of ...
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Screening for selective anticancer activity of plants from Grazalema Natural Park, Spain
Calderón Montaño, José Manuel; Martínez Sánchez, Sara María; Burgos Morón, Estefanía; Guillén Mancina, Emilio; Jiménez Alonso, Julio José; García Martín, Felipe José; Aparicio Martínez, Abelardo; López Lázaro, Miguel (Taylor & Francis, 2019-12-02)Since plants are an important source of anticancer drugs, we have carried out a random screening for selective anticancer ...
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Selective cytotoxic activity and DNA damage by an epoxyalkyl galactopyranoside
Burgos Morón, Estefanía; Pastor Carrillo, Nuria María; Orta Vázquez, Manuel Luis; Jiménez Alonso, Julio José; Vega Holm, Margarita; Vega Pérez, José Manuel; Iglesias Guerra, Fernando; Mateos Cordero, Santiago; López Lázaro, Miguel; Calderón Montaño, José Manuel (Wiley, 2018)Several clinically useful anticancer drugs selectively kill cancer cells by inducing DNA damage; the genomic instability ...
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The Cardiac Glycosides Digitoxin, Digoxin and Ouabain Induce a Potent Inhibition of Glycolysis in Lung Cancer Cells
Calderón Montaño, José Manuel; Burgos Morón, Estefanía; López Lázaro, Miguel (Biomedical Publisher, 2013)Cardiac glycosides are promising anticancer drugs. We have recently shown that the cardiac glycosides digitoxin, digoxin ...
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The Cockayne syndrome protein B is involved in the repair of 5-AZA-2′-deoxycytidine-induced DNA lesions
Burgos Morón, Estefanía; Calderón Montaño, José Manuel; Pastor Carrillo, Nuria María; Ruiz Castizo, Ángel; Domínguez García, Inmaculada; López Lázaro, Miguel; Mateos Cordero, Santiago; Orta Vázquez, Manuel Luis (Impact Journals, 2018)The Cockayne Syndrome Protein B (CSB) plays an essential role in Transcription-Coupled Nucleotide Excision Repair (TC-NER) ...