Artículo
Intracellular penetration and activity of DX-619 in human polymorphonuclear leukocytes
Autor/es | García Luque, Isabel
Ballesta, Sofía Murillo del Castillo, Concepción Perea Pérez, Evelio José Pascual Hernández, Álvaro |
Departamento | Universidad de Sevilla. Departamento de Microbiología Universidad de Sevilla. Departamento de Estomatología |
Fecha de publicación | 2006-09-01 |
Fecha de depósito | 2017-10-04 |
Publicado en |
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Resumen | The intracellular penetration and activity of DX-619 in human polymorphonuclear leukocytes have been evaluated. DX-619 reached intracellular concentrations 10 times higher than the extracellular concentrations reached. ... The intracellular penetration and activity of DX-619 in human polymorphonuclear leukocytes have been evaluated. DX-619 reached intracellular concentrations 10 times higher than the extracellular concentrations reached. Uptake was rapid, reversible, nonsaturable, and affected by environmental temperature, some metabolic inhibitors, and a soluble membrane activator. DX-619 showed intracellular activity against Staphylococcus aureus. |
Cita | García Luque, I., Ballesta, S., Murillo del Castillo, C., Perea Pérez, E.J. y Pascual Hernández, Á. (2006). Intracellular penetration and activity of DX-619 in human polymorphonuclear leukocytes. Antimicrobial Agents and Chemotherapy, 50 (9), 3173-3174. |
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