Artículo
Intracellular penetration and activity of gemifloxacin in human polymorphonuclear leukocytes
Autor/es | García Luque, Isabel
Pascual Hernández, Álvaro Joyanes, Providencia Perea Pérez, Evelio José |
Departamento | Universidad de Sevilla. Departamento de Microbiología |
Fecha de publicación | 2000-11-09 |
Fecha de depósito | 2017-09-28 |
Publicado en |
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Resumen | The intracellular penetration and activity of gemifloxacin in human polymorphonuclear leukocytes (PMN) were evaluated. Gemifloxacin reached intracellular concentrations eight times higher than extracellular concentrations. ... The intracellular penetration and activity of gemifloxacin in human polymorphonuclear leukocytes (PMN) were evaluated. Gemifloxacin reached intracellular concentrations eight times higher than extracellular concentrations. The uptake was rapid, reversible, and nonsaturable and was affected by environmental temperature, cell viability, and membrane stimuli. At therapeutic extracellular concentrations, gemifloxacin showed intracellular activity against Staphylococcus aureus. |
Cita | García Luque, I., Pascual Hernández, Á., Joyanes, P. y Perea Pérez, E.J. (2000). Intracellular penetration and activity of gemifloxacin in human polymorphonuclear leukocytes. Antimicrobial Agents and Chemotherapy, 44 (11), 3193-3195. |
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