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Listar Artículos (Química Orgánica y Farmacéutica) por autor "Mazzotta, Sarah"
Mostrando ítems 1-7 de 7
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Artículo
Antioxidant and Anti-Inflammatory Activities of Flavanones from Glycyrrhiza glabra L. (licorice) Leaf Phytocomplexes: Identification of Licoflavanone as a Modulator of NF-kB/MAPK Pathway
Frattaruolo, L.; Carullo, G; Brindisi, M; Mazzotta, Sarah; Bellissimo, L; Rago, V; Curcio, R (MDPI, 2019)Inflammation represents an adaptive response generated by injuries or harmful stimuli. Natural remedies represent an ...
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Design, synthesis and in vitro biological evaluation of a novel class of anti-adenovirus agents based on 3-amino-1,2-propanediol
Mazzotta, Sarah; Berastegui-Cabrera, Judith; Vega Holm, Margarita; García Lozano, María del Rosario; Carretero Ledesma, Marta Claudia; Aiello, Francesca; Vega Pérez, José Manuel; Pachón, Jerónimo; Iglesias Guerra, Fernando; Sánchez Céspedes, Javier (Elsevier, 2021)Nowadays there is not an effective drug for the treatment of infections caused by human adenovirus (HAdV) which supposes ...
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Design, Synthesis and In Vitro Experimental Validation of Novel TRPV4 Antagonists Inspired by Labdane Diterpenes
Mazzotta, Sarah; Carullo, Gabriele; Schiano Moriello, Aniello; Amodeo, Pietro; Marzo, Vincenzo Di; Vega Holm, Margarita; Vitale, Rosa Maria; Aiello, Francesca; Brizzi, Antonella; Petrocellis, Luciano De (MDPI, 2020)Labdane diterpenes are widespread classes of natural compounds present in variety of marine and terrestrial organisms and ...
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GPR120/FFAR4 Pharmacology: Focus on Agonists in Type 2 Diabetes Mellitus Drug Discovery
Carullo, Gabriele; Mazzotta, Sarah; Vega Holm, Margarita; Iglesias Guerra, Fernando; Vega Pérez, José Manuel; Aiello, Francesca; Brizzi, Antonella (American Chemical Society, 2021)The G-protein coupled receptors (GPCRs) activated by free fatty acids (FFAs) have emerged as new and exciting drug targets, ...
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Investigation of TNBC in vitro Antiproliferative Effects of Versatile Pirrolo[1,2-a]quinoxaline Compounds
Perri, Mariarita; Aiello, Francesca; Cione, Erika; Carullo, Gabriele; Mazzotta, Sarah; Caroleo, Maria Cristina (Frontiers Media, 2019)he triple-negative breast cancer (TNBC) is characterized by a more aggressive nature and poorer prognosis, nowadays none ...
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Piperazine-derived small molecules as potential Flaviviridae NS3 protease inhibitors. In vitro antiviral activity evaluation against Zika and Dengue viruses
García Lozano, María del Rosario; Dragoni, Filippo; Gallego, Paloma; Mazzotta, Sarah; López Gómez, Alejandro; Boccuto, Adele; Martínez-Cortés, Carlos; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Vega Pérez, José Manuel; Del Campo, José Antonio; Vicenti, Ilaria; Vega Holm, Margarita; Iglesias Guerra, Fernando (Elsevier, 2023)Since 2011 Direct Acting antivirals (DAAs) drugs targeting different non-structural (NS) viral proteins (NS3, NS5A or NS5B ...
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Repurposing Study of 4-Acyl-1-phenylaminocarbonyl-2-substituted-piperazine Derivatives as Potential Anticancer Agents-In Vitro Evaluation against Breast Cancer Cells
Guillén Mancina, Emilio; García Lozano, María del Rosario; Burgos Morón, Estefanía; Mazzotta, Sarah; Martínez Aguado, Pablo; Calderón Montaño, José Manuel; Vega Pérez, José Manuel; López Lázaro, Miguel; Iglesias Guerra, Fernando; Vega Holm, Margarita (MDPI, 2023)first_pagesettingsOrder Article Reprints Open AccessArticle Repurposing Study of 4-Acyl-1-phenylaminocarbonyl-2-substituted-piperazine ...