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Listar por autor "Bartolini, Manuela"
Mostrando ítems 1-3 de 3
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Artículo
N-1,2,3-triazole-isatin derivatives for cholinesterase and β-amyloid aggregation inhibition: A comprehensive bioassay study
Marques, Carolina S.; López López, Óscar; Bagetta, Donatella; Carreiro, Elisabete P.; Petralla, Sabrina; Bartolini, Manuela; Hoffmann, Matthias; Alcaro, Stefano; Monti, Barbara; Bolognesi, Maria Laura; Decker, Michael; Fernández-Bolaños Guzmán, José María; Burke, Anthony J. (Elsevier, 2020-05)Our goal was the evaluation of a series of N-1,2,3-triazole-isatin derivatives for multi-target activity which included ...
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Artículo
New tacrine dimers with antioxidant linkers as dual drugs: Anti-Alzheimer's and antiproliferative agents
Roldán Peña, Jesús Miguel; Alejandre Ramos, Daniel; López López, Óscar; Maya Castilla, Inés; Lagunes, Irene; Padrón, José M.; Peña Altamira, Luis Emiliano; Bartolini, Manuela; Monti, Barbara; Bolognesi, Maria L.; Fernández-Bolaños Guzmán, José María (Elsevier, 2017)We have designed a series of tacrine-based homo- and heterodimers that incorporate an antioxidant tether (selenoureido, ...
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Artículo
Tacrine-O-protected phenolics heterodimers as multitarget-directed ligands against Alzheimer's disease: Selective subnanomolar BuChE inhibitors
Roldán Peña, Jesús Miguel; Romero Real, V.; Hicke, Javier; Maya Castilla, Inés; Franconetti García, Antonio; Lagunes, Irene; Padrón, José M.; Petralla, Sabrina; Poeta, Eleonora; Naldi, Marina; Bartolini, Manuela; Monti, Barbara; Bolognesi, Maria L.; López López, Óscar; Fernández-Bolaños Guzmán, José María (Elsevier, 2019-11-01)Concerned by the devastating effects of Alzheimer's disease, and the lack of effective drugs, we have carried out the ...